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Papers of the Week


Papers: 21 Sep 2019 - 27 Sep 2019


Human Studies, Pharmacology/Drug Development


2020 Feb 01


Pain Med


21


2

Human Abuse Potential of Oral NKTR-181 in Recreational Opioid Users: A Randomized, Double-Blind, Crossover Study.

Authors

Ge X, Henningfield JE, Siddhanti S, Jobes J, Lu L, Xie S, Ziola M, Kelsh D, Vince B, Di Fonzo CJ, Tagliaferri M, Zalevsky J, Doberstein SK, Hoch U, Eldon MA
Pain Med. 2020 Feb 01; 21(2):e114-e126.
PMID: 31553457.

Abstract

To evaluate the human abuse potential, pharmacokinetics, pharmacodynamics, and safety of oral NKTR-181 (oxycodegol), a novel full mu-opioid receptor agonist, relative to oral oxycodone.